Publications
2024
Convenient syntheses of 2-acylamino-4-halothiazoles and acylated derivatives using a versatile Boc-intermediate.
Pate, S., Taujanskas, J., Wells, R., Robertson, C. M., O'Neill, P. M., & Stachulski, A. V. (2024). Convenient syntheses of 2-acylamino-4-halothiazoles and acylated derivatives using a versatile Boc-intermediate.. RSC advances, 14(38), 27894-27903. doi:10.1039/d4ra04959d
Employing transfer-dominated branching radical telomerisation (TBRT) and atom transfer radical polymerisation (ATRP) to form complex polyester-polymethacrylate branched-linear star copolymer hybrids <i>via</i> orthogonal initiation.
Dwyer, A. B., Sandy, W., Hern, F. Y., Penrhyn-Lowe, O. B., McKeating, S., Flynn, S., . . . Rannard, S. P. (2024). Employing transfer-dominated branching radical telomerisation (TBRT) and atom transfer radical polymerisation (ATRP) to form complex polyester-polymethacrylate branched-linear star copolymer hybrids <i>via</i> orthogonal initiation.. Chemical communications (Cambridge, England), 60(74), 10116-10119. doi:10.1039/d4cc02142h
2023
Thiazolide Prodrug Esters and Derived Peptides: Synthesis and Activity.
Stachulski, A. V., Rossignol, J. -F., Pate, S., Taujanskas, J., Iggo, J. A., Aerts, R., . . . O'Neill, P. M. (2023). Thiazolide Prodrug Esters and Derived Peptides: Synthesis and Activity.. ACS bio & med chem Au, 3(4), 327-334. doi:10.1021/acsbiomedchemau.2c00083
Development of Novel Thiazolides and Pyridyl Thiazolides with Improved Pharmacokinetic Properties for the Treatment of Severe Acute Respiratory Viruses and Mycobacterium Tuberculosis
Pate, S. (2023, March 6). Development of Novel Thiazolides and Pyridyl Thiazolides with Improved Pharmacokinetic Properties for the Treatment of Severe Acute Respiratory Viruses and Mycobacterium Tuberculosis.
2021
Synthesis, antiviral activity, preliminary pharmacokinetics and structural parameters of thiazolide amine salts
Stachulski, A. V., Rossignol, J. -F., Pate, S., Taujanskas, J., Robertson, C. M., Aerts, R., . . . O'Neill, P. M. (2021). Synthesis, antiviral activity, preliminary pharmacokinetics and structural parameters of thiazolide amine salts. FUTURE MEDICINAL CHEMISTRY, 13(20). doi:10.4155/fmc-2021-0055
Therapeutic Potential of Nitazoxanide: An Appropriate Choice for Repurposing versus SARS-CoV-2?
Stachulski, A. V., Taujanskas, J., Pate, S. L., Rajoli, R. K. R., Aljayyoussi, G., Pennington, S. H., . . . O'Neill, P. M. (2021). Therapeutic Potential of Nitazoxanide: An Appropriate Choice for Repurposing versus SARS-CoV-2?. ACS INFECTIOUS DISEASES, 7(6), 1317-1331. doi:10.1021/acsinfecdis.0c00478